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Patents of Ukraine

Pharmacology

  1. Utility model patent No. 66481 Ukraine, IPC (2011.01) C07D 417/00, A61K 31/425 (2006.01), A61K 31/429 (2006.01). 2,5,7-Substituted derivatives of [1,3]thiazolo[4,5-D]pyridazin-4(5H)-ones with antitumor activity // Demchenko S.A., Bobkova L.S., Demchenko A.M. – № u 201106079; Application for utility patent for Ukraine filed on May 16, 2011; Published on January 10, 2012, Bulletin No. 1.
  1. Utility model patent No. 83239 Ukraine, IPC (2013.01) C07D 417/00 A61K 31/425 (2006.01). 2-(4,5-Diphenyl-4H-[1,2,4]triazol-3-yl-sulfanyl)-N-aryl acetamides with antitumor activity // Demchenko A.M., Sukhoveyev V.V., Georgiyants V.A., Saidov N.B., Kadamov I.M., Grinevich O.Y. – No. u 2013 04229; Application for application for a patent for a new biologically active substance; Published on 27.08.2013, Bulletin No. 16.
  1. Utility model patent No. 84238 Ukraine, IPC C07D 487/04 (2006.01). Imidazole hydrochloride 3-(31,51-ditrobutyl-41-hydroxyphenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazole with antitumor properties // Demchenko A.M., Sukhoveev V.V., Moskalenko O.V., Hrynevych O.Y. – No. u 2013 05748; Application for application for patent for Ukraine filed on May 07, 2013; Published on October 10, 2013, Bulletin No. 19.
  1. Patent for invention No. 89504 Ukraine, IPC (2009), C01B 7/00, C07D 473/04 (2006.01), A61K 31/52 (2006.01), A61K 31/755 (2006.01). Adduct of 5-fluorouracil and sodium salt of diphenyl phosphoric acid for the treatment of cancer // Stefanov O.V., Sharykina N.I., Demchenko A.M., Kudriavtseva I.G., Khavych O.O., Titarenko I.P., Bobkova L.S., Sergeev V.S., Golubov M.I., Sergienko O.V. – No. a 2007 03652; Application for application for a patent for a new method of treatment of cancer.
  1. Utility model patent No. 89528 Ukraine, IPC C07D 417/00 A61P 35/00. Hydrobromides of 3-aryl-6-(4-methoxyphenyl)-7H-[1,2,4]triazolo [3,4-b][1,3,4]thiadiazine compounds with antitumor activity // Demchenko A.M., Yanchenko V.O., Sukhoveev V.V., Grinevich O.Y. – No. u 2013 13198; Application for application for 2013-11-13. Published on April 25, 2014, Bulletin No. 8.
  1. Utility model patent No. 89761 Ukraine, IPC C07D 417/00 A61P 35/00. Hydrobromides of 3-alkyl-6-(4-methoxyphenyl)-7H-[1,2,4]triazolo [3,4-b][1,3,4]thiadiazine compounds with antitumor activity // Demchenko A.M., Yanchenko V.O., Sukhoveev V.V., Grinevich O.Y. – No. u 2013 14827; Application for application for Ukraine on December 18, 2013. Published on 25.04.2014, Bulletin No. 8.
  1. Utility model patent No. 94833 Ukraine, IPC (2014.01) C07D 417/00 A61R 35/00. Substituted 7-(benzylthio)-3-tert-butyl-4H-[1,3,4]thiadiazolo[2,3-c] [1,2,4]triazine-4-ones with antitumor activity // Demchenko A.M., Yanchenko V.O., Akimenko A.O., Sukhoveev V.V. – No. u 2014 03356; Application for application for patent for Ukraine filed on April 02, 2014; Published on December 10, 2014, Bulletin No. 23.
  1. Patent for invention No. 107517 Ukraine, IPC C07D 487/04 (2006.01). Imidazole hydrochloride 3-(31,51-ditrobutyl-41-hydroxyphenyl)-6,7-dihydro-5H-pyrrolo[1,2-a]imidazole with antitumor properties // Demchenko A.M., Sukhoveev V.V., Moskalenko O.V., Hrynevych O.Y. – No. A 2013 05746; Application for application for patent for Ukraine filed on May 07, 2013; Published on January 12, 2015, Bulletin No. 1.
  1. Patent for invention No. 109814 Ukraine, IPC C07D 417/00 A61P 35/00. Hydrobromides of 3-aryl-6-(4-methoxyphenyl)-7H-[1,2,4]triazolo [3,4-b][1,3,4] thiadiazine with antitumor activity // Demchenko A.M., Yanchenko V.O., Sukhoveev V.V., Grinevich O.Y. – No. u 2013 13197; Application for application for patent for Ukraine No. 131197. Published on 12.10.2015, Bulletin No. 19.
  1. Patent for invention No. 111432 Ukraine, IPC (2016.01) A61K31/517 (2006.01), A61Z 35/00. 2-(3-Allyl-4-oxo-3,4-dihydroquinazolin-2-yl-sulfanyl)- N-(2,3-dichlorophenyl)-acetamide with antitumor effect // Sharykina N.I, Demchenko A.M., Bobkova L.S., Meshkova N.O., Kelsh Y.P., Mishchenko O.V. – No. a 2015 00282; ; Application for application for a patent for a new compound for the treatment of tumors.
  1. Utility model patent No. 116314 Ukraine, IPC (2017.01) C07D 487/04 (2006.01), A61P35/00. Hydrochloride of 2,6-Ditrobutyl-4-(6,7,8,9-tetrahydro-5H-imidazo[1,2-а]azepin-3-yl)phenol with antitumor properties // Demchenko S.A., Bobkova L.S., Demchenko A.M. – No. u 2016 13047; Application for application for patent for Ukraine on 21.14.2016; Published on 10.05.2017, Bulletin No. 9.
  1. Utility model patent No. 116804 Ukraine, IPC (2017.01) C07D 417/00. (2,3-Dihydrobenzo[1,4]dioxan-6-yl)-(3-phenyl-7H-[1,2,4]-triazolo)- [3,4-b][1,3,4]thiadiazin-6-yl) amine with antitumor activity // Demchenko A.M., Yanchenko V.O., Koval A.Y., Demenko D.A., Bobkova L.S. – No. u 2016 11805; Application for application for a patent for a new antitumor agent for the treatment of cancer.
  1. Utility model patent No. 116873 Ukraine, IPC (2017.01) C07D 417/00. 2-[4-Benzyl-5-(4′-bromophenoxymethyl)-4H-[1,2,4]triazol-3-ylsulfanyl]-N-arylacetamides with antitumor activity // Demchenko A.M., Yanchenko V.O., Saidov N.B., Georgiyants V.A., Bobkova L.S. – No. u 2016 12402; Application for application for patent for Ukraine filed on December 06, 2016; Published on June 12, 2017, Bulletin No. 11.
  1. Utility model patent No116901 Ukraine, IPC (2017.01) C07D 417/00. 2-[5-(2-Isopropyl-5-methylphenoxymethyl)-4-phenyl-4H-[1,2,4]triazol-3-yl-sulfanyl]-1-arylethanones with antitumor properties // Demchenko A.M., Dudnik A.E., Saidov N.B., Georgiyants V.A., Bobkova L.S. – No. u 2016 12799; Application for application for patent for Ukraine filed on December 15, 2016; Published on June 12, 2017, Bulletin No. 11.
  1. Utility model patent No. 116952 Ukraine, IPC (2017.01) C07D 417/00. 5,7-Diacyl-3-ethyl(cyclohexyl)-6-(4-chloro-3R-phenyl)-5H-[1,2,4]-triazolo) [3,4-b][1,3,4]Thiadiazines with antitumor activity // Demchenko A.M., Yanchenko V.O., Demchenko D.A., Bobkova L.S. – No. u 2016 13256; Application for application filed on December 26, 2016; Published on June 12, 2017, Bulletin No. 11.
  1. Utility model patent No. 117204 Ukraine, IPC (2017.01) C07D 253/065 (2006.01), C07D 295/00. N-(3,4-Dimethylphenyl)-6-morpholin-4-yl-N’-(3′-trifluoromethylphenyl)-[1,3,5]triazine-2,4-diamine with antitumor properties // Demchenko A.M., Sukhoveev V.V., Barchina O.I., Bobkova L.S. – No. u 2016 11883; Application for application for patent for Ukraine filed on November 24, 2016; Published on June 26, 2017, Bulletin No. 12.
  1. Utility model patent No. 117205 Ukraine, IPC (2017.01) C07D -417/00. 7-Phenyl-2-(1H-pyrrole-1-yl)-5H-thiazolo[4,5-d]pyridazin-4-one with antitumor properties // Demchenko S.A., Sukhoveev V.V., Bobkova L.S., Demchenko A.M. – No. u 2016 11885; Application for application for utility patent for Ukraine filed on November 24, 2016; Published on June 26, 2017, Bulletin No. 12.
  1. Utility model patent No. 117266 Ukraine, IPC (2017.01) C07D 253/065 (2006.01), C07D 295/00. 3-(2′,4′-Dichlorophenoxymethyl)-6-(4”-methoxy(or 4”-difluoromethoxyphenyl)-7H-[1,2,4]triazolo[3,4b]thiadiazines with antitumor properties // Demchenko A.M., Sukhoveev V.V., Demchenko D.A., Yanchenko V.O., Bobkova L.S. – No. u 2016 13001; Application for application for a patent for a new biological agent for the treatment of tumors.
  1. Utility model patent No. 117495 Ukraine, IPC (2017.01) C07D 417/00, A61P 35/00. 5,7-Dipropionyl-3-(4′-methoxybenzyl)-6-(4”-methoxyphenyl)-5H-[1,2,4]triazolo [4,3-b][1,3,4]Thiadiazine with antitumor activity // Demchenko A.M., Yanchenko V.O., Demchenko D.A., Bobkova L.S. – No. u 2017 00865; Application for application filed on January 31, 2017; Published on June 26, 2017, Bulletin No. 12.
  1. Utility model patent No. 117496 Ukraine, IPC (2017.01) C07D 417/00, A61K 31/425 (2006.01). 2-[5-(4-R-phenyl)-4-(meta-tolyl)-4H-[1,2,4]triazol-3-ylsulfanyl]-N-arylacetamides with antitumor properties // Demchenko A.M. – No. u 2017 00866; Application for application filed on January 31, 2017; Published on June 26, 2017, Bulletin No. 12.
  1. Utility model patent No. 117497 Ukraine, IPC (2017.01) C07D 487/04, A61P 35/00. Bromide of 3-hydroxy-1,3-bis(4′-methoxyphenyl)-2,3,5,6,7,8-hexahydroimidazo[1,2-а]pyridinium with antitumor properties // Demchenko S.A., Sukhoveev O.V., Demchenko A.M., Bobkova L.S. – No. u 2017 00868; Application for application filed on January 31, 2017; Published on June 26, 2017, Bulletin No. 12.
  1. Utility model patent No. 117545 Ukraine, IPC (2017.01) C07D 487/00, A61P 35/00. 1-Phenyl-4-aryl-5,6,7,8-tetrahydro-2,2a,8a-triazacyclopenta[c,d]azulenes with antitumor activity // Demchenko S.A., Kolesnikov O.V., Demchenko A.M., Bobkova L.S. – No. u 2017 01123; Application for application for patent for Ukraine filed on February 07, 2017; Published on June 26, 2017, Bulletin No. 12.
  1. Utility model patent No. 118179 Ukraine, IPC (2017.01) C07D 417/00. 5,7-Dipropionyl-6-(4′-cyclohexylphenyl)-5H-[1,2,4]triazolo [4,3-b][1,3,4]Thiadiazine with antitumor properties // Demchenko A.M., Yanchenko V.O., Demchenko D.A., Bobkova L.S. – No. u 2017 01375; Application for application filed on February 14, 2017; Published on July 25, 2017, Bulletin No. 14.
  1. Utility model patent No. 118189 Ukraine, IPC (2017.01) C07D 417/00. 3-(4′-methoxyphenyl)-6(4”-fluorophenyl-5,7-di-R-acyl-5H-[1,2,4]-triazolo [3,4-b][1,3,4] thiadiazines with antitumor properties, in particular, in relation to intestinal cancer cell lines // Demchenko A.M., Yanchenko V.O., Demchenko D.A., Bobkova L.S. – No. u 2017 01466; Application for application filed on February 16, 2017; Published on July 25, 2017, Bulletin No. 14.
  1. Utility model patent No. 118234 Ukraine, IPC (2017.01) C07D 417/00. 1-(2-Iso-propyl-5-methylphenoxymethyl)-3R-4-aryl-5,6,7,8-tetrahydro-2,2a,8a-triazacyclopenta[cd]azulenes with antitumor activity // Demchenko S.A, Dudnyk A.E., Bukhtiarova T.A., Demchenko A.M., Bobkova L.S. – No. u 2017 02036; Application for application for a patent for a new compound of azulenes with antitumor activity.
  1. Utility model patent No. 118683 Ukraine, IPC (2017.01) C07D 417/00. 6-(4-ethoxyphenyl)-3-(para-tolyl)-7H-[1,2,4]-triazolo [3,4-b][1,3,4]Thiadiazine with antitumor properties // Demchenko A.M., Sukhoveev V.V., Demchenko D.A., Bobkova L.S. – No. u 2017 00316; Application for application filed on January 12, 2017; Published on August 28, 2017, Bulletin No. 16.
  1. Utility model patent No. 118861 Ukraine, IPC (2017.01) C07D 487/00. 5-Benzyl-7-(furan-2-yl)-2-piperidin-1-yl-5H-thiazolo[4,5-d]-pyridazinone-4 with antitumor properties // Demchenko A.M., Sukhoveev V.V., Demchenko S.A., Sukhoveev O.V., Bobkova L.S. – No. u 2017 02991; Application for application for patent for Ukraine filed on March 30, 2017; Published on August 28, 2017, Bulletin No. 16.
  1. Utility model patent No. 120100 Ukraine, IPC (2017.01) C07D 487/00, A 61P 35/00. 4-Aryl-1-phenoxymethyl-5,6,7,8-tetrahydro-2,2a,8a-triazacyclopenta[cd]azulenes with antitumor activity // Demchenko S.A., Volochniuk D.M., Demchenko A.M., Bobkova L.S. – No. u 2017 03603; Application for application filed on April 13, 2017; Published on October 25, 2017, Bulletin No. 20.
  1. Utility model patent No. 121195 Ukraine, IPC (2017.01) C07D 487/04, A61K 31//00, A 61P 35/00. Hydrobromide of 1-(41-cyclohexylphenyl)-2-[5,6-dihydro-4H-[1,3]thiazin-2-yl)-(42-ethylphenyl)amino]ethanone with antitumor properties // Demchenko S.A., Volochniuk D.M., Bobkova L.S., Demchenko A.M. – No. u 2017 06316; Application for application for patent for Ukraine (in Ukrainian); Published on June 21, 2017; Published on November 27, 2017, Bulletin No. 22.
  1. Utility model patent No. 121779 Ukraine, IPC (2006) C07D 487/00, A 61P 35/00. 1-(21-Methoxyphenyl)aminomethyl-4-phenyl-5,6,7,8-tetrahydro-2,2a,8a-triazacyclopenta[cd] azulene with antitumor activity // Demchenko S.A., Bobkova L.S., Bukhtiarova T.A., Demchenko A.M. – No. u 2017 07644; Application for application filed on July 19, 2017; Published on December 11, 2017, Bulletin No. 23.
  1. Patent for invention No. 115644 Ukraine, IPC (2006): C07D 249/12 (2006.01), A61R 35/00. 2-[5-(4-R-phenyl)-4-(meta-tolyl)-4H-[1,2,4]triazol-3-ylsulfanyl]-N-arylacetamides with antitumor properties // Demchenko A.M. – No. a 2017 00867; Application for application for patent for Ukraine filed on January 31, 2017; Published on November 27, 2017, Bulletin No. 22.
  1. Patent for invention No. 115749 Ukraine, IPC (2006): С07D 471/04 (2006.01), С07D 487/04 (2006.01), А61Р 35/00. Pyridinium bromide 3-hydroxy-1,3-bis(4′-methoxyphenyl)-2,3,5,6,7,8-hexahydroimidazo[1,2-а]pyridinium with antitumor properties // Demchenko S.A., Sukhoveiev O.V., Demchenko A.M., Bobkova L.S. – No. u 2017 00869; Application for application filed on January 31, 2017; Published on December 11, 2017, Bulletin No. 23.
  1. Patent for invention No. 115750 Ukraine, IPC (2006): С07D 487/06 (2006.01), А61К 31/343 (2006.01), А61Р 35/00, С07С 13/52 (2006.01). 1-Phenyl-4-aryl-5,6,7,8-tetrahydro-2,2a,8a-triazacyclopenta[c,d]azulenes with antitumor activity // Demchenko S.A., Kolesnikov O.V., Demchenko A.M., Bobkova L.S. – No. a 2017 01124; Application for application for a patent for a new antitumor agent for the treatment of cancer.
  1. Utility model patent No. 123593 Ukraine, IPC (2018.01) C07D 417/00, A61K 31/425 (2006.01), A61K 31/429 (2006.01), A61P 35/04 (2006.01). 2-(7-Furan-21-yl-2-morpholin-41-yl-4-oxo-4H-thiazolo[4,5-d]pyridazin-5-yl)-N-naphthalene-1-yl-acetamide with antitumor activity // Demchenko A.M., Yarmolyuk S.M., Sharykina N.I., Bobkova L.S., Demchenko S.A., Kukharenko O.P. – No. u 2017 11183; Application for application filed on November 15, 2017; Published on February 26, 2018, Bulletin No. 4.
  1. Patent for invention No. 116424 Ukraine, IPC (2006) C07D 417/04 (2006.01), A61R 35/00, C07D 513/04 (2006.01), A61K 31/33 (2006.01). 5,7-Dipropionyl-3-(4′-methoxybenzyl)-6-(4”-methoxyphenyl)-5H-[1,2,4]triazolo [4,3-b][1,3,4]thiadiazine with antitumor activity // Demchenko A.M., Yanchenko V.O., Demchenko D.A., Bobkova L.S. – No. a 2017 00864; Application for application filed on January 31, 2017; Published on March 12, 2018, Bulletin No. 5.
  1. Patent for invention No. 116426 Ukraine, IPC (2006) C07D 417/04, A61K 31/33 (2006.01), A61R 35/00, C07D 513/04 (2006.01). 3-(4′-methoxyphenyl)-6(4”-fluorophenyl-5,7-di-R-acyl-5H-[1,2,4]-triazolo [3,4-b][1,3,4] thiadiazines with antitumor properties, in particular, in relation to intestinal cancer cell lines // Demchenko A.M., Yanchenko V.O., Demchenko D.A., Bobkova L.S. – No. a 2017 01465; Application for patent for the invention of thiadiazines, filed on February 16, 2017; Published on March 12, 2018, Bulletin No. 5.
  1. Patent for invention No. 116947 Ukraine, IPC (2006) C07D 513/04 (2006.01), A61K 31/549 (2006.01), A61R 35/00. 5,7-Diacyl-3-ethyl(cyclohexyl)-6-(4-chloro-3R-phenyl)-5H-[1,2,4]-triazolo [3,4-b][1,3,4] thiadiazines with antitumor properties // Demchenko A.M., Yanchenko V.O., Demchenko D.A., Bobkova L.S. – No. a 2016 13255; Application for application filed on December 26, 2016; Published on May 25, 2018, Bulletin No. 10.
  1. Utility model patent No. 123896 Ukraine, IPC (2006) C07D 487/00, A61P 35/00. 1-(41-Bromophenyl)-4-aryl-5,6,7,8-tetrahydro-2,2a,8a-triazacyclopenta[cd]azulenes with antitumor activity // Demchenko S.A., Artemchuk L.P., Demchenko A.M., Bobkova L.S. – No. u 2017 09889; Application for application filed on October 12, 2017; Published on March 12, 2018, Bulletin No. 5.
  1. Patent for invention No. 117404 Ukraine, IPC (2006) C07D 417/12 (2006.01), C07D 285/16 (2006.01), C07D 249/08 (2006.01), C07D 513/04 (2006.01), C07D 319/18 (2006.01), A61K 31/33 (2006.01), A61P 35/00 (2006.01). (2,3-Dihydrobenzo[1,4]dioxan-6-yl)-(3-phenyl-7H-[1,2,4]-triazolo)- [3,4-b][1,3,4]thiadiazin-6-yl) amine with antitumor activity // Demchenko A.M., Yanchenko V.O., Koval A.Y., Demchenko D.A., Bobkova L.S. – No. a 2016 11804; Application for application for a patent for a new antitumor agent for the treatment of cancer.
  1. Patent for invention No. 117406 Ukraine, IPC (2006) C07D 487/04 (2006.01), A61P35/00, A61K31/4184. Hydrochloride of 2,6-Ditrobutyl-4-(6,7,8,9-tetrahydro-5H-imidazo[1,2-а]azepin-3-yl)phenol with antitumor properties // Demchenko S.A., Bobkova L.S., Demchenko A.M. – No. a 2016 13046; Application for application for patent for Ukraine (2016), Dec. 21, 2016; Published on July 25, 2018, Bulletin No. 18.
  1. Utility model patent No. 128071 Ukraine, IPC (2006) A61K 31/381, A61K 31/498, C07D 409/12, A61P 35/00.// Ethyl-2-(quinazolin-4-yl-amino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate hydrochloride with antitumor activity in non-small cell lung cancer of humans, Demchenko A.M., Meshkova N.O., Bobkova L.S., Khairulin A.R., Mishchenko O.V., Rogozin V.V., Cherviovskyi D.O., Pendeliuk S.I., Maksiuta S.I., Bukhtiarova T.A. – № u 201804303; Application for application filed on April 19, 2018; Published on August 27, 2018, Bulletin No. 16.
  1. Utility model patent No. 129434 Ukraine, IPC (2006) A61P 35/00, C07D 417/00. 1-[6-(41-Етилфеніл)-3-метил-5-пропіоніл-5Н-[1,2,4]триазоло [3,4-b][1,3,4]thiadiazin-7-yl]-propan-1-one with antitumor properties // Demchenko A.M., Yanchenko V.O., Demchenko D.A., Bobkova L.S. – No. u 2018 05732; Application for application for the patent for Ukraine No. 2018 05732; Published on October 25, 2018, Bulletin No. 20.
  1. Patent for invention No. 118703 Ukraine, IPC (2006) C07D 417/00, A61R 35/00. 6-(4-ethoxyphenyl)-3-(para-tolyl)-7H-[1,2,4]triazolo [3,4-b][1,3,4]thiadiazine with antitumor properties // Demchenko A.M., Sukhoveev O.V., Demchenko D.A., Bobkova L.S. – No. a 2017 00318; Application for application filed on January 12, 2017; Published on February 25, 2019, Bulletin No. 4/2019.
  1. Patent for invention No. 118873 Ukraine, IPC (2006) C07D 417/00, A61K 31/425 (2006.01).//7-Phenyl-2-(1H-pyrrole-1-yl)-5H-thiazolo[4,5-d]pyridazin-4-one with antitumor properties // Demchenko S.A., Sukhoveev V.V., Bobkova L.S., Demchenko A.M. – No. a 2016 11886; Application for application on November 24, 2016; Published on March 25, 2019, Bulletin No. 6/2019.
  1. Patent for invention No. 119172 Ukraine, IPC (2017.01) C07D 249/08 (2006.01), C07D 285/16 (2006.01), C07D 417/04 (2006.01), C07D 514/04 (2006.01), A61K 31/33 (2006.01), A61R 35/00 (2006.01).// 3-(21,41-Dichlorophenoxymethyl)-6-(41-methoxy- or 41-difluoromethoxyphenyl)-7H-[1,2,4]triazolo[3,4b][1,3,4]thiadiazines with antitumor properties // Demchenko A.M, Sukhoveev V.V., Demchenko D.A., Yanchenko V.O., Bobkova L.S. – No. u 2016 12999; Application for application for a patent for a new type of thiadiazine; Declared on December 20, 2016; Published on May 10, 2019, Bulletin No. 9/2019.
  1. Patent for invention No. 119468 Ukraine, IPC (2006) C07D 255/04, A61R 35/00, A61K 31/33, A61K 31/423, C07D 249/16. Application of 1-(2-Iso-propyl-5-methylphenoxymethyl)-3R-4-aryl-5,6,7,8-tetrahydro-2,2a,8a-triazacyclopentane[cd]azulenes as compounds with antitumor activity // Demchenko S.A., Дудник А.Є., Бухтіарова Т.А., Демченко А.М., Бобкова Л.С. – № а 2017 02037; Заявл. 02.03.2017; Опубл. 25.06.2019, Бюл. № 12.
  1. Utility model patent No. 135600 Ukraine, IPC (2006) C07D 487/00, A61P 35/00, A61K 31/00.//3-R-Phenylamides of 1-(41-isopropylphenyl)-4-(42-chlorophenyl)-5,6,7,8-tetrahydro-2,4a-diazacyclopentane[c,d]azulen-2-carboxylic acid with antitumor activity against PC-3 prostate cancer cells // Demchenko S.A, Fedchenkova Y.A., Sukhoveiev V.V., Demchenko A.M. – No. u 2019 00533; Application for application on January 23, 2019; Published on July 10, 2019, Bulletin No. 13/2019.
  1. Patent for invention No. 120051 Ukraine, IPC (2017.01) C07D 251/54 (2006.01), C07D 295/00 (2006.01), A 61K 31/53 (2006.01), A 61K 31/5375 (2006.01), A 61P 35/00. The use of N-(3,4-Dimethylphenyl)-6-morpholin-4-yl-N’-(3′-trifluoromethylphenyl)-[1,3,5]triazine-2,4-diamine as an antitumor agent for the treatment of breast cancer of the MDA-MB-468 subtype // Demchenko A.M, Sukhoveiev V.V., Barchina O.I., Bobkova L.S. – No. a 2016 11884; Application for application on November 24, 2016; Published on September 25, 2019, Bulletin No. 18|2019.
  1. Utility model patent No. 136968 Ukraine, IPC (2006) C07D 487/00, A61P 35/00. [4-(41-Chlorophenyl)-5,6,7,8-tetrahydro-2,2a,8a-triazacyclopenta[cd]azulen-1-yl-methyl]-para-tolylamine, which has antitumor activity against cancer cell lines of leukemia // Demchenko S.A, Sukhoveiev V.V., Shvydko O.V., Demchenko A.M. – No. u 2019 01414; Application for application on February 12, 2019; Published on September 25, 2019, Bulletin No. 18/2019.
  1. Patent for invention No. 120182 Ukraine, IPC (2006) C07D 487/04 (2006.01), C07D 255/04 (2006.01), C07D 249/16 (2006.01), A 61K 31/33 (2006.01), A 61K 31/423 (2006.01). The use of 4-aryl-1-phenoxymethyl-5,6,7,8-tetrahydro-2,2a,8a-triazacyclopentane[cd]azulenes as compounds with antitumor activity // Demchenko S.A., Volochniuk D.M., Demchenko A.M., Bobkova L.S. – No. a 2017 03602; Application for application for a patent for Ukraine for a new antitumor agent for the treatment of cancer.
  1. Utility model patent No. 139230 Ukraine, IPC (2006) A 61K 31/5517 (2006.01), C07 D 487/04 (2006.01), C07 D 223/26 (2006.01), A 61 P 35/00. // Bromide 1-(41-methoxyphenyl)-3-(42-biphenyl)-3-hydroxy-2,5,6,7,8,8-hexahydro-3H-imidazo[1,2-а]azepinium with antitumor properties // Demchenko S.A, Fedchenkova Y.A., Sukhoveiev V.V., Demchenko A.M. – No. u 2019 06623; Application for application on June 13, 2019; Published on December 26, 2019, Bulletin No. 24/2019.
  1. Patent for invention No. 120939 Ukraine, IPC (2006) C07D 417/00, A61P 35/00, C07D 513/04 (2006.01), C07D 285/16 (2006.01), C07D 249/08 (2006.01), A61K 31/33 (2006.01). Application of 5,7-dipropionyl-6-(4′-cyclohexylphenyl)-5H-[1,2,4]triazolo [4,3-b][1,3,4]of thiadiazine as a compound with antitumor properties // Demchenko A.M., Yanchenko V.O., Demchenko D.A., Bobkova L.S. – No. a 2017 01374; Application for application for a patent for Ukraine on February 14, 2017; Published on March 10, 2020, Bulletin No. 5/20.
  1. Patent for invention No. 121172 Ukraine, IPC (2006) C07D 487/06, A61K 31/395, A61R 35/00.//3-R-Phenylamides of 1-(41-isopropylphenyl)-4-(42-chlorophenyl)-5,6,7,8-tetrahydro-2,4a-diazacyclopentane[c,d]azulen-2-carboxylic acid with antitumor activity against PC-3 prostate cancer cells // Demchenko S.A, Fedchenkova Y.A., Sukhoveiev V.V., Demchenko A.M. – No. a 2019 00686; Application for application on January 23, 2019; Published on April 10, 2020, Bulletin No. 7/2020.
  1. Patent for invention No. 121227 Ukraine, IPC (2017.01) C07D 279/06, A61K 31//54, A 61P 35/00. Application of hydrobromide 1-(41-cyclohexylphenyl)-2-[5,6-dihydro-4H-[1,3]thiazin-2-yl)-(42-ethylphenyl)amino]ethanone as a compound with antitumor properties // Demchenko S.A., Volochniuk D.M., Bobkova L.S., Demchenko A.M. – No. a 2017 06315; Application for application for a patent for a new product; Published on April 27, 2020, Bulletin No. 8/2020.
  1. Patent for invention No. 121900 Ukraine, IPC (2006) A61K 31/381, A61K 31/498, C07D 409/12, A61P 35/00. Ethyl-2-(quinazolin-4-ylamino)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate hydrochloride with antitumor activity in human non-small cell lung cancer // Sharykina N.I, Demchenko A.M., Meshkova N.O., Bobkova L.S., Khairulin A.R., Mishchenko O.V., Rogozin V.V., Cherviovskyi D.O., Pendelu S.I., Maksiuta S.V., Bukhtiarova T.A.- No. a 201804302; Application for application submitted on April 19, 2018; Published on August 10, 2020, Bulletin No. 15/2020.
  1. Patent for invention No. 123601 Ukraine, IPC (2006) C07D 487/16, A61P 35/00, A61K 31/55 Application of [4-(41-Chlorophenyl)-5,6,7,8-tetrahydro-2,2a,8a-triazacyclopentane[cd]azulen-1-yl-methyl]-para-tolylamine as an active substance with selective antitumor activity against cancer cell lines CCRF-CEM.// Demchenko SA, Sukhoveiev V.V., Shvydko O.V., Demchenko A.M. – No. a 2019 01413; Application for application on February 12, 2019; Published on April 28, 2021, Bulletin No. 17/2021.
  1. Patent for invention No. 123969 Ukraine, IPC (2006) C07D 487/04, A61K 31/55, A61P 31/00 // Bromide of 1-(41-methoxyphenyl)-3-(42-biphenyl)-3-hydroxy-2,5,6,7,8,9-hexahydro-3H-imidazo[1,2-a]azepinium with antitumor properties // Demchenko S.A., Fedchenkova Y.A., Sukhoveiev V.V., Demchenko A.M. – No. u 2019 06624; Application for application on June 13, 2019; Published on July 01, 2021, Bulletin No. 26/2021.

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